Synthesis of enantiomerically pure (2S,3S)-5,5,5-trifluoroisoleucine and (2R,3S)-5,5,5-trifluoro-allo-isoleucine

نویسندگان

  • Holger Erdbrink
  • Elisabeth K Nyakatura
  • Susanne Huhmann
  • Ulla I M Gerling
  • Dieter Lentz
  • Beate Koksch
  • Constantin Czekelius
چکیده

A practical route for the stereoselective synthesis of (2S,3S)-5,5,5-trifluoroisoleucine (L-5-F3Ile) and (2R,3S)-5,5,5-trifluoro-allo-isoleucine (D-5-F3-allo-Ile) was developed. The hydrophobicity of L-5-F3Ile was examined and it was incorporated into a model peptide via solid phase peptide synthesis to determine its α-helix propensity. The α-helix propensity of 5-F3Ile is significantly lower than Ile, but surprisingly high when compared with 4'-F3Ile.

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عنوان ژورنال:

دوره 9  شماره 

صفحات  -

تاریخ انتشار 2013